@misc{indiciaef52bf5bb479b, title = {Potent and Selective SETDB1 Covalent Negative Allosteric Modulator Reduces Methyltransferase Activity in Cells}, author = {Uguen, M. and Shell, D. J. and Silva, M. and Deng, Y. and Li, F. and Szewczyk, M. and Yang, K. and Zhao, Y. and Stashko, M. A. and Norris-Drouin, J. L. and Waybright, J. M. and Beldar, S. and Rectenwald, J. M. and Mordant, A. L. and Webb, T. S. and Herring, L. E. and Arrowsmith, C. H. and Ackloo, S. and Gygi, S. P. and McGinty, R. K. and Barsyte-Lovejoy, D. and Liu, P. and Halabelian, L. and James, L. I. and Pearce, K. H. and Frye, S. V.}, year = {2024}, doi = {10.1101/2024.09.27.615363}, url = {https://www.biorxiv.org/content/10.1101/2024.09.27.615363v1}, note = {Source identifier: 10.1101/2024.09.27.615363} }